The present invention relates to a new process for the synthesis of Colesevelam, which is used in therapy in cases of hypercholesterolemia due to low density lipoproteins. Said process comprises the reaction, in a basic environment, of polyallylamine with: i) at least one alkylating agent of formula X—(CH2)9—CH3 and at least one alkylating agent of formula Y—(CH2)6—N+ (CH3)3Z−, wherein X and Y are each independently a leaving group, and Z is a halogen; and ii) at least one crosslinking agent. The present invention also relates to the Colesevelam obtainable by the above process.


    Access

    Download


    Export, share and cite



    Title :

    DISPOSITIF DE CONTROLE POUR VEHICULE AUTOMOBILE ET PROCEDE DE COMMANDE


    Contributors:

    Publication date :

    2017-01-13


    Type of media :

    Patent


    Type of material :

    Electronic Resource


    Language :

    French


    Classification :

    IPC:    B60K Anordnung oder Einbau von Antriebseinheiten oder von Kraft- bzw. Drehmomentübertragungen in Fahrzeugen , ARRANGEMENT OR MOUNTING OF PROPULSION UNITS OR OF TRANSMISSIONS IN VEHICLES / G05G CONTROL DEVICES OR SYSTEMS INSOFAR AS CHARACTERISED BY MECHANICAL FEATURES ONLY , Steuer- oder Regelvorrichtungen oder Steuer- oder Regelsysteme gekennzeichnet ausschließlich durch mechanische Einzelheiten



    DISPOSITIF DE CONTROLE POUR VEHICULE AUTOMOBILE ET PROCEDE DE COMMANDE

    DABIC STEPHANIE / VANHELLE STEPHANE | European Patent Office | 2015

    Free access

    DISPOSITIF DE CONTROLE POUR VEHICULE AUTOMOBILE ET PROCEDE DE COMMANDE

    DABIC STÉPHANIE / TISSOT JEAN-MARC | European Patent Office | 2016

    Free access

    DISPOSITIF DE CONTROLE POUR VEHICULE AUTOMOBILE ET PROCEDE DE COMMANDE

    DABIC STEPHANIE / TISSOT JEAN MARC | European Patent Office | 2015

    Free access

    DISPOSITIF ET PROCÉDÉ DE COMMANDE POUR VÉHICULE AUTOMOBILE

    RAZUREL GUY / PITTION GILLES / BARATHON PHILIPPE et al. | European Patent Office | 2018

    Free access

    DISPOSITIF ET PROCEDE DE COMMANDE POUR VEHICULE AUTOMOBILE

    DABIC STEPHANIE / EL OUARDI NOURREDINE | European Patent Office | 2018

    Free access